| Bioactivity | NPS ALX Compound 4a is a potent and selective 5-hydroxytryptamine6 (5-HT6) receptor antagonist, with an IC50 of 7.2 nM and a Ki of 0.2 nM[1]. | ||||||||||||
| Name | NPS ALX Compound 4a | ||||||||||||
| CAS | 299433-10-6 | ||||||||||||
| Formula | C25H25N3O2S | ||||||||||||
| Molar Mass | 431.55 | ||||||||||||
| Appearance | Solid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
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| Reference | [1]. Isaac M, et al. 6-Bicyclopiperazinyl-1-arylsulfonylindoles and 6-bicyclopiperidinyl-1-arylsulfonylindolesderivatives as novel, potent, and selective 5-HT6 receptor antagonists. Bioorg Med Chem Lett. 2000 Aug 7;10(15):1719-21. |
NPS ALX Compound 4a
CAS: 299433-10-6 F: C25H25N3O2S W: 431.55
NPS ALX Compound 4a is a potent and selective 5-hydroxytryptamine6 (5-HT6) receptor antagonist, with an IC50 of 7.2 nM a
Data collection：peptidedb@qq.com
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