| Bioactivity | Milategrast is useful as cell adhesion inhibitor or cell infiltration inhibitor. Milategrast in vitro inhibites the adhesion of Jurkat cells to human fibronectin with an IC50 of <5 μM[1]. | ||||||||||||
| Name | Milategrast | ||||||||||||
| CAS | 859217-52-0 | ||||||||||||
| Formula | C24H38N2 | ||||||||||||
| Molar Mass | 354.57 | ||||||||||||
| Appearance | Solid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
| Storage |
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| Reference | [1]. Kotake, Makoto; Yoneda, Naoki; Osada, Katsunobu.Preparation of various crystal forms and salts of 1-cyclopropylmethyl-4-[2-(3,3,5,5-tetramethylcyclohexyl)phenyl]piperazine for treating or preventing various inflammatory diseases and autoimmune diseases.WO |