Bioactivity | MRS7935 (compound 15) is an A1AR positive allosteric modulator (PAM) with an EC50 of approximately 2 μM[1]. |
Target | EC50: 2 μM (Adenosine receptor A1AR) |
Name | MRS7935 |
Formula | C24H20ClF2NOS |
Molar Mass | 443.94 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Oliva P et al. 2-Amino-5-arylethynyl-thiophen-3-yl-(phenyl) methanones as A1 Adenosine Receptor Positive Allosteric Modulators[J]. ACS Medicinal Chemistry Letters, 2023. |