| Bioactivity | MRS1186 is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist, with a Ki of 7.66 nM. |
| Target | Ki: 7.66 nM (hA3AR). |
| Invitro | MRS1186 (compound 2d) is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist, with a Ki of 7.66 nM[1]. |
| Name | MRS1186 |
| CAS | 183721-03-1 |
| Formula | C16H12ClN5O2 |
| Molar Mass | 341.75 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Tafi A, et al. Pharmacophore based receptor modeling: the case of adenosine A3 receptor antagonists. An approach to the optimization of protein models. J Med Chem. 2006 Jul 13;49(14):4085-97. |