Bioactivity | MRGPRX4 agonist-1 (compound 30d) is a selective agonist of MRGPRX4 with EC50s of 11.2 nM and 30.0 nM in Ca2+ and β-arrestin experiments, respectively[1]. |
Target | MRGPRX4 |
Name | MRGPRX4 agonist-1 |
CAS | 2768131-22-0 |
Formula | C21H25N4O6P |
Molar Mass | 460.42 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Marx D et al. Discovery of Potent Agonists for the Predominant Variant of the Orphan MAS-Related G Protein-Coupled Receptor X4 (MRGPRX4). J Med Chem. 2023 Nov 15. |