| Bioactivity | MRGPRX1 agonist 2 (compound 1a) is a potent Mas-related G protein-coupled receptor X1 (MRGPRX1) positive allosteric modulator with an EC50 value of 0.48 μM. MRGPRX1 agonist 2 can be used for researching neuropathic pain[1]. |
| Target | EC50: 0.48 μM (MRGPRX1) |
| Name | MRGPRX1 agonist 2 |
| CAS | 302952-43-8 |
| Formula | C15H14N2OS |
| Molar Mass | 270.35 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Berhane I, et al. Thieno[2,3-d]pyrimidine-Based Positive Allosteric Modulators of Human Mas-Related G Protein-Coupled Receptor X1 (MRGPRX1). J Med Chem. 2022;65(4):3218-3228. |
MRGPRX1 agonist 2
CAS: 302952-43-8 F: C15H14N2OS W: 270.35
MRGPRX1 agonist 2 (compound 1a) is a potent Mas-related G protein-coupled receptor X1 (MRGPRX1) positive allosteric modu
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