| Bioactivity | MRGPRX1 agonist 1 is a highly potent agonist of MRGPRX1 (Mas-related G-protein-coupled receptor X1), with an EC50 of 50 nM, and is inactive on MRGPRC11. Analgesic effect[1]. | ||||||||||||
| Target | EC50: 50 nM (MRGPRX1) | ||||||||||||
| Name | MRGPRX1 agonist 1 | ||||||||||||
| CAS | 2377379-39-8 | ||||||||||||
| Formula | C23H21N3O4S | ||||||||||||
| Molar Mass | 435.50 | ||||||||||||
| Appearance | Solid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
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| Reference | [1]. Prchalová E, et al. Discovery of Benzamidine- and 1-Aminoisoquinoline-Based Human MAS-Related G-Protein-Coupled Receptor X1 (MRGPRX1) Agonists. J Med Chem. 2019 Sep 26;62(18):8631-8641. |
MRGPRX1 agonist 1
CAS: 2377379-39-8 F: C23H21N3O4S W: 435.50
MRGPRX1 agonist 1 is a highly potent agonist of MRGPRX1 (Mas-related G-protein-coupled receptor X1), with an EC50 of 50
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