| Bioactivity | MMSET-IN-1 is a multiple myeloma SET domain (MMSET, aka NSD2/WHSC1) inhibitor against SETD2 and MMSET with IC50s of 0.49 and 3.3 μM, respectively. MMSET-IN-1 has a Kd of 1.6 μM for MMSET[1]. |
| Target | IC50: 0.49 μM (SETD2), 3.3 μM (MMSET)Kd: 1.6 μM |
| Name | MMSET-IN-1 |
| CAS | 1998139-29-9 |
| Formula | C18H29N7O5 |
| Molar Mass | 423.47 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Tisi D, et al. Structure of the Epigenetic Oncogene MMSET and Inhibition by N-Alkyl Sinefungin Derivatives. ACS Chem Biol. 2016 Nov 18;11(11):3093-3105. |
MMSET-IN-1
CAS: 1998139-29-9 F: C18H29N7O5 W: 423.47
MMSET-IN-1 is a multiple myeloma SET domain (MMSET, aka NSD2/WHSC1) inhibitor against SETD2 and MMSET with IC50s of 0.49
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