| Bioactivity | MM 54 (compound 5) is a competitive antagonist at APJ, with an IC50 of 93 nM. MM 54 behaves as a potent and selective inhibitor of apelin binding and APLNR activation[1][2]. | ||||||
| Invitro | MM 54 inhibits more than 95% of apelin binding to APLNR at the dose of 10 µM[2]. | ||||||
| Name | MM 54 | ||||||
| CAS | 1313027-43-8 | ||||||
| Shortening | CRPRLCKHCRPRLC (Disulfide bridge:Cys1-Cys6; Cys9-Cys14) | ||||||
| Formula | C70H121N29O15S4 | ||||||
| Molar Mass | 1737.17 | ||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||
| Storage | Sealed storage, away from moisture and light, under nitrogen
*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light, under nitrogen) |
MM 54
CAS: 1313027-43-8 F: C70H121N29O15S4 W: 1737.17
MM 54 (compound 5) is a competitive antagonist at APJ, with an IC50 of 93 nM. MM 54 behaves as a potent and selective in
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