| Bioactivity | MM 07 is a biased apelin receptor agonist, with a KD of 300 nM in CHO-K1 cells and a KD of 172 nM in human heart. | ||||||
| Invitro | MM 07 competes with nanomolar affinities for binding of [Glp65,Nle75,Tyr77] [125I]apelin-13 to human apelin receptors in CHO-K1 cells (KD, 300 nM) and human heart (KD, 172 nM, n=3)[1]. | ||||||
| Name | MM 07 | ||||||
| CAS | 1876450-21-3 | ||||||
| Sequence | Cys-Arg-Pro-Arg-Leu-Cys-His-Lys-Gly-Pro-Met-Pro-Phe (Disulfide bridge:Cys1-Cys6) | ||||||
| Shortening | CRPRLCHKGPMPF (Disulfide bridge:Cys1-Cys6) | ||||||
| Formula | C67H106N22O14S3 | ||||||
| Molar Mass | 1539.89 | ||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||
| Storage | Sealed storage, away from moisture
*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture) |