| Bioactivity | MCHR1 antagonist 1 is a selective antagonist of melanin concentrating hormone-1 (MCH1) receptor, with a Kb of 1 nM and a Ki of 4 nM at human MCH1, and may be used to reduce the body mass. |
| Target | Kb: 1 nM (Human MCH1)Ki: 4 nM (Human MCH1) |
| Invitro | MCHR1 antagonist 1 shows potent activities against melanin concentrating hormone-1 receptor, but less potent against human MCH1, NPY1, NPY5, GALR1, GALR2, GALR3, and rat 5HT2C receptors, with Kis of >50000 nM[1]. |
| Name | MCHR1 antagonist 1 |
| CAS | 391610-37-0 |
| Formula | C28H33F2N5O5 |
| Molar Mass | 557.59 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Selective melanin concentrating hormone-1 (MCH1) receptor antagonists and uses thereof. US 20030069261 A1 |
MCHR1 antagonist 1
CAS: 391610-37-0 F: C28H33F2N5O5 W: 557.59
MCHR1 antagonist 1 is a selective antagonist of melanin concentrating hormone-1 (MCH1) receptor, with a Kb of 1 nM and a
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