Bioactivity | M1/M2/M4 muscarinic agonist 3 (compound 45) is a muscarinic mAChR M1/M2/M4 agonist with EC50s of 3.2 nM, 32 nM and 1.7 nM, respectively[1]. |
Target | EC50: 3.2 nM (M1 muscarinic receptor), 32 nM (M2 muscarinic receptor), 1.7 nM (M4 muscarinic receptor) |
Name | M1/M2/M4 muscarinic agonist 3 |
CAS | 2640109-28-8 |
Formula | C23H31FN2O3 |
Molar Mass | 402.50 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Thomson C G et al. Transaminases Provide Key Chiral Building Blocks for the Synthesis of Selective M1/M4 Agonists[J]. ACS Medicinal Chemistry Letters, 2023. |