| Bioactivity | Lofexidine-d4 is deuterium labeled Lofexidine (hydrochloride). Lofexidine (hydrochloride) is a selective α2-receptor agonist, commonly used to alleviate the physical symptoms of heroin and other types of opioid withdrawal[1][2][3]. |
| CAS | 78302-26-8 |
| Formula | C11H8D4Cl2N2O |
| Molar Mass | 263.16 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019 Feb;53(2):211-216. [2]. Vartak AP, et al. The preclinical discovery of lofexidine for the treatment of opiate addiction. Expert Opin Drug Discov. 2014 Nov;9(11):1371-7. [3]. Gish EC, et al. Lofexidine, an {alpha}2-receptor agonist for opioid detoxification. Ann Pharmacother. 2010 Feb;44(2):343-51. |
Lofexidine-d4
CAS: 78302-26-8 F: C11H8D4Cl2N2O W: 263.16
Lofexidine-d4 is deuterium labeled Lofexidine (hydrochloride). Lofexidine (hydrochloride) is a selective α2-receptor ag
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