| Bioactivity | LXQ-87 is an oral allosteric inhibitor of PTP1B with an IC50 of 1.061 μM, showing hypoglycemic activity. LXQ-87 alleviates insulin resistance and promotes cellular glucose uptake, making it useful for research on type 2 diabetes[1]. |
| CAS | 2524718-73-6 |
| Formula | C23H18Br2O5 |
| Molar Mass | 534.19 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Chenxia Gao, et al. Allosteric inhibition of PTP1B by bromocatechol-chalcone derivatives. Eur J Med Chem. 2025 Jan 15:282:117053. |