Bioactivity | LPAR1 antagonist 2 (example 76) is an LPAR1 antagonist with an average IC50 of 130 nM[1]. |
Target | Mean IC50: 130 nM (LPAR1) |
CAS | 1664336-46-2 |
Formula | C23H20ClNO4 |
Molar Mass | 409.86 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Preparation of amide derivatives as lysophosphatidic acid receptor antagonists. World Intellectual Property Organization, et al. World Intellectual Property Organization, WO2015025164 A1 2015-02-26. |