| Bioactivity | LK 204-545 is a potent and highly selective β1-adrenoceptor antagonist. LK 204-545 is promising for research of cardiovascular diseases[1]. |
| CAS | 83068-69-3 |
| Formula | C25H32N4O6 |
| Molar Mass | 484.54 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Louis S N S, et al. LK 204-545, a highly selective β1-adrenoceptor antagonist at human β-adrenoceptors[J]. European journal of pharmacology, 1999, 367(2-3): 431-435. [2]. Mistry SN, et al. Synthesis and in vitro and in vivo characterization of highly β1-selective β-adrenoceptor partial agonists. J Med Chem. 2013 May 23;56(10):3852-65. |