| Bioactivity | LBG20304 (compound 2s) is a ligand for the homologous GluK5 receptor (IC50: 432 nM), more than 40-fold selective over the homologous GluK1-3 isoforms. Low doses of LBG20304 (10 μM), it exhibits low agonist activity in neuronal slices (rat)[1]. |
| Target | IC50: 432 nM (GluK5) |
| Formula | C19H18N4O5 |
| Molar Mass | 382.37 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Domoic Acid as a Lead for the Discovery of the First Selective Ligand for Kainate Receptor Subtype 5 (GluK5) |