| Bioactivity | L-659837 is a NK2 receptor antagonist, and can antagonize GR 64349 (HY-P1278)-induced contraction. L-659837 can be used for study of urinary bladder disorders[1]. |
| CAS | 125989-10-8 |
| Sequence | Cyclo(Gln-Trp-Phe-{(R)Gly(ANC-2)}-Leu-Met) |
| Shortening | Cyclo(QWF-{(R)Gly(ANC-2)}-LM) |
| Formula | C40H52N8O7S |
| Molar Mass | 788.96 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Palea S, et al. Pharmacological characterization of tachykinin NK2 receptors on isolated human urinary bladder, prostatic urethra and prostate. J Pharmacol Exp Ther. 1996;277(2):700-705. |