| Bioactivity | KSK94 is a high-affinity histamine H3 receptor antagonist, with Kis of 7.9, 2958, 75.2 nM for H3 receptor, sigma-1, sigma-2 receptor respectively. KSK94 can be used for research of nociceptive and neuropathic pain[1]. |
| Target | 7.9, 2958, 75.2 nM (H3 receptor, sigma-1, sigma-2 receptor) |
| Name | KSK94 |
| CAS | 2566716-07-0 |
| Formula | C25H26N4O |
| Molar Mass | 398.50 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Szczepańska K, et al. Dual Piperidine-Based Histamine H3 and Sigma-1 Receptor Ligands in the Treatment of Nociceptive and Neuropathic Pain. J Med Chem. 2023 Jul 27;66(14):9658-9683. |