| Bioactivity | KFM19 is a potent, selective Adenosine receptor (A1-receptor) antagonist, with an IC50 of 50 nM. | ||||||||||||
| Target | IC50: 50 nM (Adenosine receptor) | ||||||||||||
| Name | KFM19 | ||||||||||||
| CAS | 133058-72-7 | ||||||||||||
| Formula | C16H22N4O3 | ||||||||||||
| Molar Mass | 318.37 | ||||||||||||
| Appearance | Solid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
| Storage |
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| Reference | [1]. W.D. Bechtel, et al. KFM 19 antagonizes the adenosine-induced inhibition of electrically evoked acetylcholine release. Eur Neuropsychopharmacol. Sep. 1993, 3(3), Page 433 |