| Bioactivity | K-(D-1-Nal)-FwLL-NH2 TFA is a high affinity and potent ghrelin receptor inverse agonist (Ki values are 4.9 and 31 nM in COS7 and HEK293T cells, respectively). K-(D-1-Nal)-FwLL-NH2 blocks ghrelin receptor-mediated Gq- and G13-dependent signaling pathways. |
| Name | K-(D-1-Nal)-FwLL-NH2 TFA |
| Sequence | Lys-{Nal}-Phe-Trp-Leu-Leu-NH2 |
| Shortening | K{Nal}FWLL-NH2 |
| Formula | C53H68F3N9O8 |
| Molar Mass | 1016.16 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |