| Bioactivity | JTP-117968, a novel selective glucocorticoid receptor modulator (a non-steroidal SGRM, IC50 of 6.8 nM), exhibits improved transrepression/transactivation dissociation[1]. |
| Invitro | JTP-117968 has partial TR activity, but exhibits extremely low TA activity[1]. |
| Name | JTP-117968 |
| CAS | 2250132-99-9 |
| Formula | C31H31F3N2O2 |
| Molar Mass | 520.59 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Takafumi Kurimoto, et al. JTP-117968, a novel selective glucocorticoid receptor modulator, exhibits improved transrepression/transactivation dissociation. Eur J Pharmacol. 2017 May 15;803:179-186. |
JTP-117968
CAS: 2250132-99-9 F: C31H31F3N2O2 W: 520.59
JTP-117968, a novel selective glucocorticoid receptor modulator (a non-steroidal SGRM, IC50 of 6.8 nM), exhibits improve
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