Bioactivity | Idelalisib-d5 is a deuterium labeled Idelalisib. Idelalisib is a highly selective and orally bioavailable p110δ inhibitor[1]. | ||||||||||||
Target | P110δ inhibitor | ||||||||||||
Name | Idelalisib-d5 | ||||||||||||
CAS | 1830330-31-8 | ||||||||||||
Formula | C22H13D5FN7O | ||||||||||||
Molar Mass | 420.45 | ||||||||||||
Appearance | Solid | ||||||||||||
Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
Storage |
|
||||||||||||
Reference | [1]. Lannutti BJ, et al. CAL-101, a p110delta selective phosphatidylinositol-3-kinase inhibitor for the treatment of B-cell malignancies, inhibits PI3K signaling and cellular viability. Blood, 2011, 117(2), 591-594. |