| Bioactivity | IRE1α kinase-IN-4 (compound 6) is a potent IRE1α inhibitor with an Ki of 140 nM. IRE1α kinase-IN-4 is the ATP-competitive ligands of IRE1α[1]. |
| Target | Ki: 140 nM (IRE1α) |
| Name | IRE1α kinase-IN-4 |
| CAS | 2771006-45-0 |
| Formula | C29H31N7O2 |
| Molar Mass | 509.60 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Feldman HC, et al. ATP-competitive partial antagonists of the IRE1α RNase segregate outputs of the UPR. Nat Chem Biol. 2021 Nov;17(11):1148-1156. |
IRE1α kinase-IN-4
CAS: 2771006-45-0 F: C29H31N7O2 W: 509.60
IRE1α kinase-IN-4 (compound 6) is a potent IRE1α inhibitor with an Ki of 140 nM. IRE1α kinase-IN-4 is the ATP-competi
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