| Bioactivity | IRAP-IN-1 (compound 3) is a potent and selective insulin regulated aminopeptidase (IRAP) inhibitor with an IC50 value of 157 nM[1]. |
| Target | IC50: 157 nM (IRAP) |
| Formula | C26H28N6O3 |
| Molar Mass | 472.54 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Anastasia Mpakali, et al.Stabilization of the open conformation of Insulin-Regulated Aminopeptidase by a novel substrate-selective small molecule inhibitor. Biorxiv, 2024. |