IDH1 Inhibitor 2_product_DataBase

CAS: 2244895-42-7 F: C26H22N4O W: 406.48

IDH1 Inhibitor 2 (compound 13) is a potent wild-type IDH1 inhibitor via a direct covalent modification of His315, with a

This product is for research use only, not for human use. We do not sell to patients.

Bioactivity	IDH1 Inhibitor 2 (compound 13) is a potent wild-type IDH1 inhibitor via a direct covalent modification of His315, with an IC50 of 110 nM[1].
Target	IC50: 110 nM (IDH1).
Name	IDH1 Inhibitor 2
CAS	2244895-42-7
Formula	C26H22N4O
Molar Mass	406.48
Transport	Room temperature in continental US; may vary elsewhere.
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.
Reference	[1]. Jakob CG, et al. Novel Modes of Inhibition of Wild-Type Isocitrate Dehydrogenase 1 (IDH1): Direct Covalent Modification of His315. J Med Chem. 2018 Aug 9;61(15):6647-6657.

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