| Bioactivity | ICI 174864 is a highly selective, potent δ-receptor antagonist. ICI 174864 is equipotent with naloxone and can not reverse the effect of the μ-agonist [D-Ala2, MePhe4, Gly-Ol5]enkephalin or the κ-agonist tifluadom[1]. |
| Name | ICI 174864 |
| CAS | 89352-67-0 |
| Sequence | {N,N-diallyl}-Tyr-{Aib}-Phe-Leu |
| Shortening | {N,N-diallyl}-Y-{Aib}-FL |
| Formula | C34H46N4O6 |
| Molar Mass | 606.75 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. R Cotton, et, al. ICI 174864: a highly selective antagonist for the opioid delta-receptor. Eur J Pharmacol. 1984, 97,3. |