| Bioactivity | HPSE1-IN-2 (compound 2) is a Heparanase-1 (HPSE1) inhibitor that also inhibits exo-β-d-glucuronidase (GUSβ) and glucocerebrosidase (GBA) activity[1]. |
| Target | Heparanase-1 (HPSE1), exo-β-d-glucuronidase (GUSβ) and glucocerebrosidase (GBA) |
| Name | HPSE1-IN-2 |
| CAS | 2876926-27-9 |
| Formula | C23H24N2O6 |
| Molar Mass | 424.45 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Imai Y et al. Discovery of a novel tetrahydroimidazo [1, 2-a] pyridine-5-carboxylic acid derivative as a potent and selective heparanase-1 inhibitor utilizing an improved synthetic approach[J]. Bioorganic & Medicinal Chemistry Letters, 2023: 129543. |