| Bioactivity | HPK1-IN-44 (Compound 1) is an inhibitor of HPK1 (IC50=0.1 nM (40 μM ATP))[1]. |
| Invitro | HPK1-IN-44 的细胞学活性结果分别为 IC50=120.88 nM (pSLP76); EC50=3.67 nM (IL-2 release)[1]。 MCE has not independently confirmed the accuracy of these methods. They are for reference only. 0 --> HPK1-IN-44 相关抗体: |
| Formula | C29H26ClN5O2 |
| Molar Mass | 512.00 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Guanglong S et al. HPK1 inhibitor, preparation method therefor, and use thereof.World Intellectual Property Organization, WO2024061345 A1 2024-03-28 |