Bioactivity | H4R antagonist 3 (Example 18) is a histamine-4 receptor antagonist with an EC50 of <10 mM. H4R antagonist 3 can be used for the research of prevention of inflammatory, autoimmune, allergic, and ocular diseases[1]. |
Target | EC50: <10 mM (histamine-4 receptor) |
Name | H4R antagonist 3 |
CAS | 1003091-20-0 |
Formula | C19H21ClN4S |
Molar Mass | 372.91 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Allen J. Borchardt, et al. Aminopyrimidine inhibitors of histamine receptors for the treatment of disease. Patent US20100063047A1. |