Bioactivity | H2L5186303 is a potent and selective LPA2 receptor (lysophosphatidic acid 2 receptor) antagonist with an IC50 of 9 nM[1]. | ||||||||||||
Name | H2L5186303 | ||||||||||||
CAS | 139262-76-3 | ||||||||||||
Formula | C26H20N2O8 | ||||||||||||
Molar Mass | 488.45 | ||||||||||||
Appearance | Solid | ||||||||||||
Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
Storage |
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Reference | [1]. Fells JI, et al. Structure-based drug design identifies novel LPA3 antagonists. Bioorg Med Chem. 2009 Nov 1;17(21):7457-64. |