Bioactivity | GSTP1-1 inhibitor 1 (compound 6b) is an irreversible, long-acting, glutathione S-transferase inhibitor with an IC50 of 21 μM targeting GSTP1-1 . GSTP1-1 is a key tumor suppressor target, and GSTP1-1 inhibitor 1 has potential anticancer activity[1]. |
Target | IC50: 21 μM (GSTP1-1) |
Name | GSTP1-1 inhibitor 1 |
CAS | 3829-23-0 |
Formula | C6H3ClFNO4S |
Molar Mass | 239.61 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Shishido Y, et al. A Covalent Inhibitor for Glutathione S‐Transferase Pi (GSTP1‐1) in Human Cells[J]. ChemBioChem, 2019, 20(7): 900-905. |