Bioactivity | GSTO1-IN-2 (Compound B-9) is a dual covalent inhibitor of GSTO1/BTK with IC50 values of 441 nM and 6.2 nM respectively[1]. |
Target | IC50: 441 nM (GSTO1).IC50: 6.2 nM (BTK). |
CAS | 3020776-77-3 |
Formula | C30H24N8O2 |
Molar Mass | 528.56 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Liu Y, et al. Proteome-wide Ligand and Target Discovery by Using Strain-Enabled Cyclopropane Electrophiles[J]. Journal of the American Chemical Society, 2024. |