| Bioactivity | GST-IN-1 (compound 16) is a glutathione S-transferase (GST) inhibitor with IC50s of 1.55 μM (sjGST) and 2.02 μM (hGSTM2), respectively. |
| Target | IC50: 1.55 μM (sjGST) and 2.02 μM (hGSTM2) |
| Name | GST-IN-1 |
| Formula | C29H20Cl2N6O3S |
| Molar Mass | 603.48 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Wen X, Zhang M, Duan Z, Suo Y, Lu W, Jin R, Mu B, Li K, Zhang X, Meng L, Hong Y, Wang X, Hu H, Zhu J, Song W, Shen A, Lu X. Discovery, SAR Study of GST Inhibitors from a Novel Quinazolin-4(1H)-one Focused DNA-Encoded Library. J Med Chem. 2023 Aug 24;66(16):11118-11132. |