| Bioactivity | GSK3004774 is a potent, nonabsorbable agonist of CaSR, with an pEC50 of 7.3, 6.6 and 6.5 for human, mouse and rat CaSR, respectively. GSK3004774 shows an EC50 of 50 nM for human CaSR[1]. |
| Name | GSK3004774 |
| CAS | 2138814-32-9 |
| Formula | C32H40N4O3 |
| Molar Mass | 528.69 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Sparks SM, et al. Identification of potent, nonabsorbable agonists of the calcium-sensing receptor for GI-specific administration. Bioorg Med Chem Lett. 2017 Oct 15;27(20):4673-4677. |
GSK3004774
CAS: 2138814-32-9 F: C32H40N4O3 W: 528.69
GSK3004774 is a potent, nonabsorbable agonist of CaSR, with an pEC50 of 7.3, 6.6 and 6.5 for human, mouse and rat CaSR,
Data collection：peptidedb@qq.com
This product is for research use only, not for human use. We do not sell to patients.