| Bioactivity | GSK2973980A is a potent and selective Acyl-CoA:diacylglycerol acyltransferase 1 (DGAT1) inhibitor with an IC50 of 3 nM. |
| Target | IC50: 3 nM (DGAT1) |
| Name | GSK2973980A |
| CAS | 2219321-25-0 |
| Formula | C25H19F5N4O4 |
| Molar Mass | 534.43 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Cheung M, et al. Discovery of Tetralones as Potent and Selective Inhibitors of Acyl-CoA:Diacylglycerol Acyltransferase 1. ACS Med Chem Lett. 2018 Jan 16;9(2):103-108. |
GSK2973980A
CAS: 2219321-25-0 F: C25H19F5N4O4 W: 534.43
GSK2973980A is a potent and selective Acyl-CoA:diacylglycerol acyltransferase 1 (DGAT1) inhibitor with an IC50 of 3 nM.
Data collection：peptidedb@qq.com
This product is for research use only, not for human use. We do not sell to patients.