Bioactivity | GSK2606414 is a cell-permeable and orally available protein kinase R-like endoplasmic reticulum (ER) kinase (PERK) inhibitor with an IC50 of 0.4 nM. | ||||||||||||
Invitro | GSK2606414 inhibits PERK activation in cells[1]. | ||||||||||||
Name | GSK2606414 | ||||||||||||
CAS | 1337531-36-8 | ||||||||||||
Formula | C24H20F3N5O | ||||||||||||
Molar Mass | 451.44 | ||||||||||||
Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
Storage |
|