| Bioactivity | GS-462808 is an oral active late sodium current inhibitor (Late INai) of the cardiac Nav1.5 channel with the IC50 of 1.33 μM. GS-462808 can be used for study of arrhythmia[1]. |
| CAS | 1354198-41-6 |
| Formula | C17H12F3N5O3 |
| Molar Mass | 391.30 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Koltun DO, et al. Discovery of triazolopyridinone GS-462808, a late sodium current inhibitor (Late INai) of the cardiac Nav1.5 channel with improved efficacy and potency relative to ranolazine. Bioorg Med Chem Lett. 2016;26(13):3207-3211. |
GS-462808
CAS: 1354198-41-6 F: C17H12F3N5O3 W: 391.30
GS-462808 is an oral active late sodium current inhibitor (Late INai) of the cardiac Nav1.5 channelwith the IC50 of 1.33
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