| Bioactivity | GRL018-21 is a potent and highly selective G protein-coupled receptor kinase 5 (GRK5) inhibitor with an IC50 value of 10 nM[1]. |
| Name | GRL018-21 |
| Formula | C30H25FN4O5 |
| Molar Mass | 540.54 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Chen Y, et al. Development of a new class of potent and highly selective G protein-coupled receptor kinase 5 inhibitors and structural insight from crystal structures of inhibitor complexes[J]. European Journal of Medicinal Chemistry, 2023: 115931. |