| Bioactivity | GRK2 Inhibitor 1 (methyl 5-[2-(5-nitro-2-furyl)vinyl]-2-furoate) is a GRK2 (β-ARK1) inhibitor[1]. | ||||||||||||
| Name | GRK2 Inhibitor 1 | ||||||||||||
| CAS | 24269-96-3 | ||||||||||||
| Formula | C12H9NO6 | ||||||||||||
| Molar Mass | 263.20 | ||||||||||||
| Appearance | Solid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
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| Reference | [1]. Nimitvilai S, et al. Reversal of dopamine D2 agonist-induced inhibition of ventral tegmental area neurons by Gq-linked neurotransmitters is dependent on protein kinase C, G protein-coupled receptor kinase, and dynamin. J Pharmacol Exp Ther. 2013 Jan;344(1 |