| Bioactivity | GR65630 is a potent and selective 5-hydroxytryptamine (5-HT) type 3 receptor antagonist. GR65630 can be used to study the expression patterns of 5-HT3 receptors in different brain regions and their possible functions in the central nervous system. GR65630 and its radiolabeled form [3H]GR65630 can be used to study the distribution, density and affinity of the receptors[1]. |
| CAS | 113140-33-3 |
| Formula | C16H17N3O |
| Molar Mass | 267.33 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Kilpatrick G J, et al. Binding of the 5-HT3 ligand,[3H] GR65630, to rat area postrema, vagus nerve and the brains of several species[J]. European journal of pharmacology, 1989, 159(2): 157-164. |