| Bioactivity | GR 94800 is a potent and selective NK2 receptor peptide antagonist, with pKB values of 9.6, 6.4 and 6.0 for NK2, NK1 and NK3 receptors, respectively[1][2]. |
| Invitro | Responses to EFS (15 Hz) were significantly reduced by the NK2 receptor antagonist GR 94800 (1 μM) either alone or in combination with the NK1 antagonist (1 μM)[3]. |
| Name | GR 94800 |
| CAS | 141636-65-9 |
| Shortening | Bz-AA-{D-Trp}-F-{D-Pro}-P-{Nle}-NH2 |
| Formula | C49H61N9O8 |
| Molar Mass | 904.06 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |