Bioactivity | GR 196429 is a melatonin receptor agonist with some selectivity for the MT1 subtype. GR 196429 produces both sleep-promoting effects and alterations of circadian rhythm, as well as stimulating melatonin release in mice[1]. |
Name | GR 196429 |
CAS | 170729-12-1 |
Formula | C14H18N2O2 |
Molar Mass | 246.30 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. I J Beresford, et al. Pharmacological characterisation of melatonin mt1 receptor-mediated stimulation of [35S]-GTPgammaS binding. Biochem Pharmacol. 1998 Nov 1;56(9):1167-74. |