| Bioactivity | GR 128107 is a competitive melatonin receptor antagonist (pKi: 9.6)[1]. |
| Name | GR 128107 |
| CAS | 190328-44-0 |
| Formula | C16H20N2O2 |
| Molar Mass | 272.34 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Dubocovich ML, et al. Melatonin receptor antagonists that differentiate between the human Mel1a and Mel1b recombinant subtypes are used to assess the pharmacological profile of the rabbit retina ML1 presynaptic heteroreceptor. Naunyn Schmiedebergs Arch Pharmacol. 1997 Mar;355(3):365-75. |