| Bioactivity | GPR81 agonist 2 (compound 1) is a potent GPR81 agonist with EC50 values of 0.023, 0.123 µM for hGPR81, hGPR109A, respectively[1]. |
| Target | EC50: 0.023 (hGPR81); 0.123 µM (hGPR109A) |
| Name | GPR81 agonist 2 |
| CAS | 1143024-28-5 |
| Formula | C26H27ClN6O5S2 |
| Molar Mass | 603.11 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Davidsson Ö, et al. Identification of novel GPR81 agonist lead series for target biology evaluation. Bioorg Med Chem Lett. 2020 Feb 15;30(4):126953. |