Bioactivity | GPR55 agonist 4 (Compound 28) is a GPR55 agonist (EC50: 131 nM, and 1.41 nM for hGPR55 and rGPR55). GPR55 agonist 4 induces β-arrestin recruitment to human GPR55[1]. |
Name | GPR55 agonist 4 |
Formula | C19H16FN5O2 |
Molar Mass | 365.36 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Hewer RC, et al. Discovery and Characterization of Novel CNS-Penetrant GPR55 Agonists. J Med Chem. 2023 Sep 28;66(18):12858-12876. |