Bioactivity | GPR41 modulator 1 (compound 10ak) is a potent GPR41 modulator with an EC50 value of 0.679 µM. GPR41 modulator 1 shows agonistic modulator activity[1]. |
Target | EC50: 0.679 µM (GPR41) |
Invitro | GPR41 modulator 1 (compound 10ak) (1 µM) 可降低 HEK293 细胞中丙酸(10 mM)诱导的 cAMP 水平[1]。 MCE has not independently confirmed the accuracy of these methods. They are for reference only. 0 --> GPR41 modulator 1 相关抗体: |
Formula | C28H24F2N2O3 |
Molar Mass | 474.50 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Inuki S, et al. Structure-activity relationship studies of tetrahydroquinolone derivatives as GPR41 modulators. Bioorg Med Chem Lett. 2024 Jul 15;107:129758. |