| Bioactivity | GPR40 agonist 1 is a potent and novel GPR40 full agonist with an EC50 of 2 nM and 17 nM for hGPR40 and rGPR40, respectively. |
| Target | EC50: 2 nM (hGPR40), 17 nM (rGPR40) |
| Name | GPR40 agonist 1 |
| CAS | 1853982-41-8 |
| Formula | C27H30FN3O4 |
| Molar Mass | 479.54 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Meegalla SK, et al. Discovery of a novel potent GPR40 full agonist. Bioorg Med Chem Lett. 2018 Feb 15;28(4):720-726. |