| Bioactivity | GPR35 agonist 2 (compound 11) is a potent agonist of GPR35, with EC50s of 26 and 3.2 nM in the β-arrestin and Ca2+ release assay, respectively[1]. |
| Target | EC50: 26 nM (human GPR35 in β-arrestin), 3.2 nM (human GPR35 in Ca2+ release assay) |
| Name | GPR35 agonist 2 |
| CAS | 494191-73-0 |
| Formula | C17H11FN2O3S |
| Molar Mass | 342.34 |
| Appearance | Solid |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | 4°C, protect from light *In solvent : -80°C, 6 months; -20°C, 1 month (protect from light) |
| Reference | [1]. Thimm D, et, al. 6-Bromo-8-(4-[(3)H]methoxybenzamido)-4-oxo-4H-chromene-2-carboxylic Acid: a powerful tool for studying orphan G protein-coupled receptor GPR35. J Med Chem. 2013 Sep 12; 56(17): 7084-99. |
GPR35 agonist 2
CAS: 494191-73-0 F: C17H11FN2O3S W: 342.34
GPR35 agonist 2 (compound 11) is a potent agonist of GPR35, with EC50s of 26 and 3.2 nM in the β-arrestin and Ca2+ rele
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