Bioactivity | GPR183-IN-1 (compound 15) is a potent and orally activity GPR183 inhibitor. GPR183-IN-1 inhibits Ca2+ mobilization with an IC50 value of 39.97 nM. GPR183-IN-1 has the potential for the research of cancer, autoimmune diseases, pain, and osteoporosis[1]. |
In Vivo | 药代动力学分析[1].Parameters |
CAS | 2924063-70-5 |
Formula | C16H19BrN2O2 |
Molar Mass | 351.24 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. JianFei Xi, et al. Compounds and their use as GPR183 inhibitors. CN118201911A. |